 Other References: |
"Substitution and Additons in the Heterocyclic Rings of Nucleic Acid Bases and Their Derivative--§, Sub-section 1 (Halogenation)," in Ch. 5 of Organic Chemistry of Nucleic Acids, Part B, Kochetkov et al. (Russian eds.), Haigh et al. (English translator & eds.), Plenum Press, New York, NY, 1972, only pp. 269-275 supplied.
Goodman, "Chemical Synthese and Transformations of Nucleosides,", Ch. 2 in Basic Principles in Nucleic Acid Chemistry, vol. 1, Ts'o (ed.), Academic Press, New York, NY, 1974, only pp. 146-152 and 202 supplied.
Robins et al., "A Direct Synthesis of 5-Fluorocytosine and Its Nucleosides Using Trifluoromethyl Hypofluorite," J. Chem. Soc., Part D(Chem. Comm.), (1), pp. 18-19, (Jan. 5, 1972).
Jorge R. Barrio, et al., Regioselective Fluorination of Substituted Guanines with Dilute F2 : A Facile Entry to 8-Fluoroguanine Derivates, J. Org. Chem., 1996, 61, 6084-6085., Issue No. 18, Sep. 6, 1996.
(2 pages)
Cited by 2 patents
[ISI abstract]
Jorge R. Barrio, et al., "Elemental Fluorine to 8-Fluoropurines in One Step" J. American Chem. Soc., 1996, 118, 10408-10411., Issue No. 43, Oct. 30 1996.
(4 pages)
Cited by 3 patents
[ISI abstract]
William Braker, et al., "Matheson Gas Data Book," Matheson Gas Products, East Rutherford, N.J. 1971,. pp. 261-265 only.
Sono, M., et al., "Functionalization Including Fluorination of Nitrogen-Containing Compounds Using Electrochemical Oxidation," Chem. Pharm. Bull., vol. 44, No. 6, pp. 1141-1145 (Jun. 1996).
(5 pages)
Cited by 3 patents
[ISI abstract]
Jorge R. Barrio, et al., A Direct Method for the Preparation of 2-Hydroxyethoxymethly Derivatives of Guanine, Adenine, and Cytosine, J. Med. Chem, 1980, 23, 572-574, issue No. 5.
(3 pages)
Cited by 10 patents
Ratsep, P., et al., "Introduction of Fluorine Into the C8 Position Of Purine Nucleosides," Nucleosides & Nucleotides, 1990, 9(2), pp. 197-204.
(8 pages)
Cited by 2 patents
Pross, A., "A General Approach to Organic Reactivity: The Configuration Mixing Model," Advances in Physical Organic Chemistry, 1985, vol. 21, pp. 99-198.
(98 pages)
Cited by 2 patents
Lacan, G., et al., "Fluorination of (E)-β-(Fluoromethylene)-m-Tyrosine: Regioselective Synthesis of 4-Fluoro-(E)-β-(Fluoromethylene)-m-Tyrosine," J. Org. Chem., 1995, vol. 60, No. 1, pp. 227-234.
(8 pages)
Cited by 2 patents
[ISI abstract]
Barrio, Jorge R., et al., "A Direct Method for the Preparation of 2-Hydroxyethoxymethyl Derivatives of Guanine, Adenine, and Cytosine", J. Med. Chem., 1980, vol. 23, No. 5, pp. 572-574.
(3 pages)
Cited by 10 patents
Satyamurthy, N., et al., "Making 18 F radiotracers for medical research," Chemtech, Mar. 1994, pp. 25-32.
(8 pages)
Cited by 2 patents
[ISI abstract]
Coenen, H.H., et al., "Regiospecific Aromatic Fluorodemetallation of Group IVb Metalloarenes Using Elemental Flourine or Acetyle Hypofluorite," Journal of Fluorine Chemistry, 1987, vol. 36, p. 63.
(13 pages)
Cited by 3 patents
Walsh, C., "Fluorinated Substrate Analogs: Routes of Metabolism and Selective Toxicity," In Advances in Enzymology: Meister, A. Ed: John Wiley and Sons: New York, 1983: vol. 55 pp. 197-289.
(93 pages)
Cited by 2 patents
Welch, J. T., "Advances in the Prepration of Biologically Active Organofluorine Compounds," Tetrahedron, 1987, vol. 43, No. 14, pp. 3123-3197.
(75 pages)
Cited by 6 patents
Welch, J. T., Ed., American Chem. Soc.: Washington, DC "Selective Fluorination in Organic and Bioorganic Chemistry," American Chemical Society, Apr. 22, 1990.
Barnett, W.C., CRC Critical Reviews in Biochemistry, vol. 15, Issue 3, pp. 210-213.
Marquez, Victor E., et al., "Acid-Stable 2'-Fluoro Purine Dideoxynucleosides as Active Agents against HIV," J. Med. Chem., 1990, vol. 33, No. 3, pp. 978-985.
(8 pages)
Cited by 15 patents
Robins, M. J., et al., "Nucleic acid related compounds. 34. Non-aqueous diazotization with tert-butyl nitrite. Introduction of fluorine, chlorine, and bromine at C-2 of purine nucleosides," Can. J. Chem., 1981, vol. 59, pp. 2608-2611.
(4 pages)
Cited by 7 patents
Montgomery, J. A., et al., "Synthesis and Biological Evaluation of 2-Fluoro-8-azaadenosine and Related Compounds1," J. Med. Chem., 1983, vol. 26, No. 10, pp. 1483-1489.
(7 pages)
Cited by 2 patents
Secrist III, J.A., et al., "2-Fluoroformycin and 2-Aminoformycin. Synthesis and Biological Activity," J. Med. Chem., 1985, vol. 28, No. 11, pp. 1740-1742.
(3 pages)
Cited by 4 patents
Secrist III, J. A., et al., "Synthesis and Biochemical Properties of 8-Amino-6-fluoro-9-β-D-ribofuranosyl-9H-purine,"J. Med. Chem., 1986, vol. 29, No. 10, pp. 2029.-2074.
Secrist III, J.A., "Synthesis and Biological Evaluations of Certain 2-Halo-2'-Substituted Derivatives of 9-β-D-Arabinofuranosyladenine," J. Med. Chem., 1988, vol. 31, No. 2, pp. 405-410.
(6 pages)
Cited by 6 patents
Robins, M. J., et al., "Nucleic Acid Related Compounds. III. A Facile Synthesis of 5-Fluorouracil Bases and Nucleosides by Direct Fluorination," Journal of the American Chemical Society, vol. 93, 1971, pp. 5277-5278 (Oct. 6, 1971).
Robins, M. J., et al., "Nucleic Aacid Related Compounds. 21. Direct Fluorination of Uracil and Cytosine Bases and Nucleosides Using Trifluoromethyl Hypoflourite. Mechanism, Stereochemistry, and Synthetic Applications," Journal of the American Chemical Society, 1976, vol. 98, p. 7381.(Nov. 10, 1976).
(10 pages)
Cited by 2 patents
Gerstenberger, M.R.C., et al., "Methods of Fluorination in Organic Chemistry," Angew: Chem. Int. Ed. Engl., 1981, vol. 20, p. 647.
(21 pages)
Cited by 9 patents
Beaman, A. G., et al., "The Direct Conversion of Chloropurines to Fluoropurines," J. Org. Chem., 1963, vol. 28, pp. 2310-2313.
Naik, S. R., et al., "A Novel Route to 3(5)-Fluoro-1,2,4-triazoles and 8-Fluoropurines by Displacement of the Nitro Group," J. Org. Chem., 1973, vol. 38, No. 25, pp. 4353-4354.
(2 pages)
Cited by 3 patents
Ikehara, M., et al., "Studies of Nucleosides and Nucleotides. XLIX. Synthesis of 8-Fluoroadenosine," Chem. Pharm. Bull., 1971, vol. 19, pp. 104-109. Issue No. 1.
Kobayashi, Y., et al., "Synthesis of 2',3',5'-Tris-O-acetyle-8-fluoroadenosine," J.C.S. Chem. Comm., 1976, pp. 430-431.
(2 pages)
Cited by 2 patents
Sono, M., et al., "Functionalisation Including Fluorination of Caffeine, Guanosine Tetraacetate, and Uridine Triacetate using Electrochemical Oxidation," Tetrahedron Letters, 1994, vol. 35, No. 49, pp. 9237-9238.
(2 pages)
Cited by 2 patents
[ISI abstract]
Rozen, S., "The formation of the C-F bond: the last twelve years," Supplement D2: The chemistry of halides, pseudo-halides and azides, Patai, S. et al. Eds: John Wiley and Sons: Chichester, U.K. 1995; Chapter 12, pp. 629-708.
Rozen, S., et al., "Remote and Selective Electrophilic Fluorinations at the Carbon-Hyrogen Single Bond," J. Am. Chem. Soc., 1980, vol. 102, No. 22, pp. 6860-6861.
(2 pages)
Cited by 2 patents
Shiue, C., et al., "A New Improved Synthesis of 2-Deoxy-2-[18 F]Fluoro-D-Glucose from 18 F-Labeled Acetyl Hypofluorite," The Journal of Nuclear Medicine, 1982, vol. 23, No. 10, pp. 899-903.
(5 pages)
Cited by 5 patents
Kosower, E. M., et al., "Bimanes. 21. syn-(Methyl,fluoro)bimane, Formation via Acetyl Hypofluorite," J. Org. Chem., 1985, vol. 50, No. 21, pp. 4152-4154.
(3 pages)
Cited by 2 patents
Luxen, A., et al., "Electrophilic And Nucleophilic Approaches to the Synthesis of 3-Fluorodiazepam," Journal of Fluorine Chemistry, 1987, 36, pp. 83-92.
(10 pages)
Cited by 2 patents
Bryce, M. R., et al., "Electrophilic fluorination of tin and mercury derivatives as a route to fluoroaromatics," Bulletin De La Societe Chimique De France, 1986. No. 6, pp. 930-932.
(3 pages)
Cited by 3 patents
Fused Pyrimides, Brown, D.J. Ed., Part II, Purines; Meister, J.H. Ed.; Wiley-Interscience: New York, 1971, Chapter V, pp. 136.-201.
Stolarski, R., et al., "Comparison Of Theoretical and Experimental Approaches To Determination of Conformation of Nucleosides About The Glycosidic Bond," Biochimica et Biophysica Acta, 1980, 610, pp. 1-19.
(19 pages)
Cited by 2 patents
Silverman, R.B. in Mechanism-Based Enzyme Inactivation: Chemistry and Enzymology; CRC Press, Inc.: Boca Raton, FL, 1988; vol. 1, pp. 59-93.
Mario Ikehara and Tohikazu Fukui, Studies of Nucleosides and Nucleotides. LVIII*.Deamination of Adenosine Analogs with Calf Intestine Adenosine Deaminase, Biochemical et Biophysica Acta, vol. 338, 1974; 512-519.
(8 pages)
Cited by 2 patents
|
Nominate this for the Gallery...
